Enzalutamide 40 mg
Price range: $1,943.50 through $5,577.26
| Quantity Value | Price | Quantity | Add To Cart |
|---|---|---|---|
| 28 Capsule/s | $1,943.50 |
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| 56 Capsule/s | $3,785.78 |
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| 84 Capsule/s | $5,577.26 |
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SKU : N/A
Category : Anti Cancer , Life Saving , Prostate Cancer
Enzalutamide 40 mg is used to treat prostate cancer by blocking androgen receptors, slowing cancer growth and improving survival in advanced or metastatic cases.
Enzalutamide 40 mg Capsules are an advanced oral medication used in the treatment of prostate cancer. Recognized for their targeted and effective anti-cancer properties, these capsules play a crucial role in managing various stages of prostate cancer, particularly castration-resistant and metastatic types. This medication is classified as an androgen receptor inhibitor and functions by blocking the effects of androgens (male hormones) that fuel the growth of prostate cancer cells. As part of a broader treatment regimen, Enzalutamide 40 mg has significantly improved outcomes and extended survival in many patients.
Prostate cancer remains one of the most prevalent malignancies in men. As the disease progresses, it often becomes resistant to standard hormonal therapies. Enzalutamide is specifically formulated to address this resistance, offering a powerful solution when traditional approaches fail.
Composition and Formulation
Each capsule of Enzalutamide 40 mg contains 40 mg of the active ingredient Enzalutamide. The medication is presented in a soft gelatin capsule for ease of oral consumption. Additional pharmaceutical excipients are included to ensure proper delivery, absorption, and bioavailability in the body. The formulation is designed to offer consistent performance across a wide range of patients, regardless of age or stage of disease.
Mechanism of Action
Enzalutamide belongs to a class of medications known as androgen receptor inhibitors. Androgens, including testosterone and dihydrotestosterone, play a central role in the growth and survival of prostate cancer cells. Unlike traditional antiandrogens that merely block the binding of these hormones, Enzalutamide inhibits multiple steps in the androgen receptor signaling pathway:
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Prevents binding of androgens to the androgen receptor.
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Inhibits nuclear translocation of the androgen receptor.
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Blocks DNA binding of the androgen receptor complex.
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Disrupts transcription of androgen-responsive genes.
By interfering with this hormonal pathway at several levels, Enzalutamide delivers a more comprehensive and sustained anti-cancer effect than earlier-generation antiandrogens.
Indications
Enzalutamide 40 mg Capsules are indicated for:
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Metastatic Castration-Resistant Prostate Cancer (mCRPC)
For patients whose disease progresses despite surgical or medical castration. -
Non-Metastatic Castration-Resistant Prostate Cancer (nmCRPC)
For patients who have not yet developed metastases but are no longer responding to hormonal therapy. -
Metastatic Castration-Sensitive Prostate Cancer (mCSPC)
In combination with androgen deprivation therapy (ADT) for patients newly diagnosed with metastatic disease.
These indications allow Enzalutamide to serve patients at different phases of their cancer journey, helping extend survival and improve quality of life.
Dosage and Administration
The standard adult dose of Enzalutamide is 160 mg per day, typically administered as four 40 mg capsules taken once daily, at the same time each day. The capsules can be taken with or without food, but consistency in timing is recommended to maintain stable blood levels.
Swallow capsules whole with water. Do not crush, chew, or dissolve the capsules, as this may affect the drug’s integrity and efficacy.
Missed Dose: If a dose is missed, it should be taken as soon as possible on the same day. If a full day has passed, skip the missed dose and resume normal dosing the next day. Do not double the dose to make up for a missed one.
Benefits of Enzalutamide 40 mg Capsules
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Extended Survival: Enzalutamide has shown significant improvements in overall survival for patients with advanced prostate cancer.
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Non-Invasive Treatment: Unlike chemotherapy, Enzalutamide offers an oral route of administration, avoiding invasive procedures and hospital stays.
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Delays Disease Progression: It can slow the spread of cancer, particularly in non-metastatic castration-resistant cases.
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Improved Quality of Life: By controlling symptoms such as bone pain and urinary complications, Enzalutamide enhances patient comfort.
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No Need for Steroids: Unlike some alternative treatments, it does not require concurrent steroid use, reducing the risk of steroid-associated side effects.
Side Effects
As with any potent medication, Enzalutamide may cause side effects in some individuals. Common side effects include:
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Fatigue
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Hot flashes
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Back pain
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Hypertension
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Headaches
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Diarrhea
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Joint pain
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Dizziness
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Weight loss
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Swelling in hands or feet
Less common but more serious side effects include:
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Seizures
Rare but potentially severe; caution is advised in patients with a history of epilepsy or brain injury. -
Falls and Fractures
Especially in elderly patients or those with bone metastases. -
Cognitive Effects
Confusion, memory issues, or trouble concentrating may occur in some patients.
Patients experiencing any severe or persistent symptoms should consult their healthcare provider immediately.
Precautions
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Pre-existing Conditions: Use with caution in patients with a history of seizures, cardiovascular disease, or liver impairment.
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Pregnancy and Breastfeeding: This medication is not intended for use in women. It may harm unborn babies and is contraindicated during pregnancy.
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Drug Interactions: Enzalutamide is known to interact with medications metabolized by CYP enzymes in the liver. Inform your doctor of all medications and supplements you are taking.
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Driving and Operating Machinery: Due to the potential for dizziness, fatigue, or seizures, patients should avoid hazardous tasks until they know how the drug affects them.
Drug Interactions
Enzalutamide may interact with a wide variety of other drugs, including:
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Anticoagulants (e.g., warfarin)
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Anticonvulsants (e.g., phenytoin)
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Antiarrhythmics (e.g., amiodarone)
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Immunosuppressants (e.g., tacrolimus)
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St. John’s Wort and other herbal supplements
It is critical to inform your physician or pharmacist of all prescription and non-prescription medications you are currently using.
Storage Instructions
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Store at room temperature between 20°C to 25°C (68°F to 77°F).
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Keep the container tightly closed and away from moisture and direct sunlight.
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Do not freeze the capsules.
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Keep out of reach of children and pets.
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Dispose of unused medication in accordance with local pharmacy regulations.
FAQs
1. How long will I need to take Enzalutamide 40 mg?
Treatment duration depends on individual response, disease progression, and tolerability. It may be used long-term in some cases.
2. Can I stop treatment if I feel better?
No. Stopping the medication abruptly can result in a rapid return of cancer symptoms. Always consult your doctor before making changes.
3. Can I drink alcohol while on Enzalutamide 40 mg?
Moderate alcohol use may be acceptable for some, but alcohol can increase dizziness or fatigue. Discuss with your healthcare provider.
4. Is monitoring required during treatment?
Yes. Regular blood tests and imaging may be necessary to track disease progression and monitor liver function.
Conclusion
Enzalutamide 40 mg Capsules offer a powerful and flexible solution for men battling prostate cancer. With its ability to delay disease progression, extend survival, and maintain quality of life, it represents one of the most effective oral therapies available today. By targeting the androgen receptor pathway more comprehensively than older treatments, Enzalutamide provides new hope to patients living with advanced prostate cancer.
When used responsibly and under the supervision of a qualified healthcare provider, Enzalutamide can play a transformative role in modern prostate cancer care.
| Quantity Value |
28 Capsule/s ,56 Capsule/s ,84 Capsule/s |
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